Assay
PGDB_AS000212
System: cell_basedCell line: MM.1R
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 5-10 | nM | - | — | - | - | MM.1R | WO2024032689A1 | PGDB_A014790 | PGDB_C002489 | PGDB_AS000212 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MM.1R | WO2024032689A1 | PGDB_A019885 | PGDB_C002495 | PGDB_AS000212 | View | |
| IC50 | - | <= | 5 | nM | - | — | - | - | MM.1R | WO2024032689A1 | PGDB_A038125 | PGDB_C002491 | PGDB_AS000212 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | MM.1R | WO2024032689A1 | PGDB_A042442 | PGDB_C002488 | PGDB_AS000212 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | MM.1R | WO2024032689A1 | PGDB_A065017 | PGDB_C002487 | PGDB_AS000212 | View |