Assay

PGDB_AS000280

System: cell_basedTarget: NEK7
Assay context summary

Assay context

212 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetNEK7
E3CRBN
Technologyluminescence
Activity compounds and values

Activity records

212 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020387
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A007257PGDB_C020387PGDB_AS000280View
2D structure for PGDB_C020391
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A008355PGDB_C020391PGDB_AS000280View
2D structure for PGDB_C020304
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A008777PGDB_C020304PGDB_AS000280View
2D structure for PGDB_C020327
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A008869PGDB_C020327PGDB_AS000280View
2D structure for PGDB_C016406
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A008917PGDB_C016406PGDB_AS000280View
2D structure for PGDB_C020368
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A008974PGDB_C020368PGDB_AS000280View
2D structure for PGDB_C020444
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A008981PGDB_C020444PGDB_AS000280View
2D structure for PGDB_C016351
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A008984PGDB_C016351PGDB_AS000280View
2D structure for PGDB_C020416
DC50->1000nM-—NEK7CRBN-WO2025024521A1PGDB_A009359PGDB_C020416PGDB_AS000280View
2D structure for PGDB_C020427
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A009472PGDB_C020427PGDB_AS000280View
2D structure for PGDB_C020346
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A009982PGDB_C020346PGDB_AS000280View
2D structure for PGDB_C020367
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A010018PGDB_C020367PGDB_AS000280View
2D structure for PGDB_C020388
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A010066PGDB_C020388PGDB_AS000280View
2D structure for PGDB_C020193
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A010482PGDB_C020193PGDB_AS000280View
2D structure for PGDB_C020414
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A010538PGDB_C020414PGDB_AS000280View
2D structure for PGDB_C020450
DC50-=100-1000nM-—NEK7CRBN-WO2025024521A1PGDB_A010707PGDB_C020450PGDB_AS000280View
2D structure for PGDB_C020294
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A010855PGDB_C020294PGDB_AS000280View
2D structure for PGDB_C020324
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A011046PGDB_C020324PGDB_AS000280View
2D structure for PGDB_C020317
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A011284PGDB_C020317PGDB_AS000280View
2D structure for PGDB_C020332
DC50-<100nM-—NEK7CRBN-WO2025024521A1PGDB_A012137PGDB_C020332PGDB_AS000280View
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