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SIMM · NJU
Assay
PGDB_AS000334
System: cell_based
Target: IKZF1
Cell line: 293GT
Assay context summary
Assay context
150 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF1
E3
CRBN
Cell line
293GT
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
150 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A007300
PGDB_C022706
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A007513
PGDB_C022690
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A008258
PGDB_C022766
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A009118
PGDB_C022671
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A009766
PGDB_C022704
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A010542
PGDB_C022673
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A011713
PGDB_C022725
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A011966
PGDB_C022724
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013441
PGDB_C022771
PGDB_AS000334
View
EC50
-
>
50.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013626
PGDB_C022640
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013850
PGDB_C022755
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A015794
PGDB_C022751
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A016186
PGDB_C022705
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A016212
PGDB_C022659
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A016541
PGDB_C022731
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A016663
PGDB_C022683
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A016696
PGDB_C022765
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A017112
PGDB_C022723
PGDB_AS000334
View
EC50
-
>
50.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A017368
PGDB_C022643
PGDB_AS000334
View
EC50
-
>
30.0
uM
-
—
-
-
293GT
CN111051298A
PGDB_A018106
PGDB_C022707
PGDB_AS000334
View