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Cc1ccc2sc(-c3ccc(CN4CCC(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)nc2c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A016212 | PGDB_C022659 | PGDB_AS000334 | View | |
| % Degradation | - | = | 65.0 | % | 10 uM | 24 h | - | - | 293GT | CN111051298A | PGDB_A050687 | PGDB_C022659 | PGDB_AS002112 | View | |
| EC50 | - | = | 0.12 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A054096 | PGDB_C022659 | PGDB_AS001169 | View | |
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A059380 | PGDB_C022659 | PGDB_AS002316 | View |