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SIMM · NJU
Assay
PGDB_AS000440
System: biochemical
Target: BTRC | FBXW11 | SKP1
Assay context summary
Assay context
193 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
BTRC | FBXW11 | SKP1
E3
BTRC | FBXW11 | SKP1
Activity compounds and values
Activity records
193 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007293
PGDB_C020826
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007599
PGDB_C020863
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A007958
PGDB_C020870
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009867
PGDB_C020906
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A010646
PGDB_C020873
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A011458
PGDB_C020893
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A011474
PGDB_C020914
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A011504
PGDB_C020981
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012052
PGDB_C020791
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012151
PGDB_C020976
PGDB_AS000440
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012259
PGDB_C020987
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012559
PGDB_C020866
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012727
PGDB_C020874
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012769
PGDB_C020835
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A012784
PGDB_C020796
PGDB_AS000440
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013344
PGDB_C020833
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013479
PGDB_C020850
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013594
PGDB_C020960
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A013816
PGDB_C020944
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A014177
PGDB_C020905
PGDB_AS000440
View