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COc1cc2c(cc1N1CCCC3(CC3)C1=O)CN(C(=O)c1c(Sc3c(Cl)cccc3Cl)cc(C(F)(F)F)[nH]c1=O)C2CC#N| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | < | 1 | uM | - | — | CTNNB1 | BTRC | FBXW11 | - | WO2025179005A1 | PGDB_A012559 | PGDB_C020866 | PGDB_AS000440 | View | |
| EC50 | - | < | 1 | uM | - | — | NFE2L2 | BTRC | FBXW11 | - | WO2025179005A1 | PGDB_A040496 | PGDB_C020866 | PGDB_AS002080 | View | |
| EC50 | - | < | 1 | uM | - | — | NFE2L2 | BTRC | FBXW11 | - | WO2025179005A1 | PGDB_A058986 | PGDB_C020866 | PGDB_AS002080 | View | |
| EC50 | - | < | 1 | uM | - | — | CTNNB1 | BTRC | FBXW11 | - | WO2025179005A1 | PGDB_A076861 | PGDB_C020866 | PGDB_AS000440 | View |