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SIMM · NJU
Assay
PGDB_AS000645
System: cell_based
Target: IKZF1
Cell line: HEK293
Assay context summary
Assay context
140 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
IKZF1
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
140 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
44
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A007700
PGDB_C005897
PGDB_AS000645
View
Dmax
-
=
27
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A007762
PGDB_C005979
PGDB_AS000645
View
Dmax
-
=
95
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A007890
PGDB_C005887
PGDB_AS000645
View
Dmax
-
=
88
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A007912
PGDB_C005956
PGDB_AS000645
View
Dmax
-
=
55
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008074
PGDB_C005976
PGDB_AS000645
View
Dmax
-
=
36
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008625
PGDB_C005918
PGDB_AS000645
View
Dmax
-
=
51
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A010846
PGDB_C005999
PGDB_AS000645
View
Dmax
-
=
71
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A011706
PGDB_C005883
PGDB_AS000645
View
Dmax
-
=
30
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A011943
PGDB_C005917
PGDB_AS000645
View
Dmax
-
=
23
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A012350
PGDB_C005923
PGDB_AS000645
View
Dmax
-
=
97
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A013056
PGDB_C005965
PGDB_AS000645
View
Dmax
-
=
67
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A013566
PGDB_C005879
PGDB_AS000645
View
Dmax
-
=
35
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A015291
PGDB_C005881
PGDB_AS000645
View
Dmax
-
=
93
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A015426
PGDB_C005912
PGDB_AS000645
View
Dmax
-
=
95
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A015787
PGDB_C005871
PGDB_AS000645
View
Dmax
-
=
30
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A016370
PGDB_C005944
PGDB_AS000645
View
Dmax
-
=
42
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A016744
PGDB_C005994
PGDB_AS000645
View
Dmax
-
=
97
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A016859
PGDB_C005986
PGDB_AS000645
View
Dmax
-
=
50
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A017211
PGDB_C006010
PGDB_AS000645
View
Dmax
-
=
86
%
-
24 h
IKZF1
-
HEK293
AU2022419982A1
PGDB_A017256
PGDB_C005890
PGDB_AS000645
View