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SIMM · NJU
Assay
PGDB_AS000646
System: cell_based
Target: GSPT1
Cell line: NB4
Assay context summary
Assay context
32 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
GSPT1
E3
Not specified
Cell line
NB4
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
32 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
44
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A007077
PGDB_C003334
PGDB_AS000646
View
Dmax
-
=
74
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A013511
PGDB_C003347
PGDB_AS000646
View
Dmax
-
=
86
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A016049
PGDB_C003344
PGDB_AS000646
View
Dmax
-
=
22
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A017887
PGDB_C003336
PGDB_AS000646
View
Dmax
-
=
128
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A020146
PGDB_C003340
PGDB_AS000646
View
Dmax
-
=
68
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A021669
PGDB_C003346
PGDB_AS000646
View
Dmax
-
=
91
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A022573
PGDB_C003333
PGDB_AS000646
View
Dmax
-
=
117
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A022622
PGDB_C003353
PGDB_AS000646
View
Dmax
-
=
129
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A026702
PGDB_C003350
PGDB_AS000646
View
Dmax
-
=
106
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A027445
PGDB_C003341
PGDB_AS000646
View
Dmax
-
=
125
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A028740
PGDB_C003357
PGDB_AS000646
View
Dmax
-
=
122
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A029306
PGDB_C003335
PGDB_AS000646
View
Dmax
-
=
118
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A030469
PGDB_C003338
PGDB_AS000646
View
Dmax
-
=
105
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A030540
PGDB_C003362
PGDB_AS000646
View
Dmax
-
=
107
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A033104
PGDB_C003351
PGDB_AS000646
View
Dmax
-
=
103
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A043783
PGDB_C003364
PGDB_AS000646
View
Dmax
-
=
96
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A045063
PGDB_C003361
PGDB_AS000646
View
Dmax
-
=
119
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A045476
PGDB_C003356
PGDB_AS000646
View
Dmax
-
=
119
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A046957
PGDB_C003352
PGDB_AS000646
View
Dmax
-
=
109
%
5 mM
4 h
GSPT1
-
NB4
WO2025146129A1
PGDB_A052676
PGDB_C003337
PGDB_AS000646
View