Assay

PGDB_AS000657

System: cell_basedTarget: VAV1
Assay context summary

Assay context

77 activity records
Assay family% Degradation
Systemcell_based
ReadoutDmax
TargetVAV1
E3Not specified
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C032056
Dmax-=96.9%0.02 nM-VAV1--WO2026119120A1PGDB_A000096PGDB_C032056PGDB_AS000657View
2D structure for PGDB_C009245
Dmax-=90.8%0.02 nM-VAV1--WO2026119120A1PGDB_A000255PGDB_C009245PGDB_AS000657View
2D structure for PGDB_C032004
Dmax-=92.5%0.02 nM-VAV1--WO2026119120A1PGDB_A000317PGDB_C032004PGDB_AS000657View
2D structure for PGDB_C032002
Dmax-=94.8%0.02 nM-VAV1--WO2026119120A1PGDB_A000378PGDB_C032002PGDB_AS000657View
2D structure for PGDB_C032063
Dmax-=95.8%0.02 nM-VAV1--WO2026119120A1PGDB_A000385PGDB_C032063PGDB_AS000657View
2D structure for PGDB_C032067
Dmax-=95.7%0.02 nM-VAV1--WO2026119120A1PGDB_A000566PGDB_C032067PGDB_AS000657View
2D structure for PGDB_C032026
Dmax-=91.9%0.02 nM-VAV1--WO2026119120A1PGDB_A000572PGDB_C032026PGDB_AS000657View
2D structure for PGDB_C032069
Dmax-=94.8%0.02 nM-VAV1--WO2026119120A1PGDB_A000687PGDB_C032069PGDB_AS000657View
2D structure for PGDB_C032044
Dmax-=96.5%0.02 nM-VAV1--WO2026119120A1PGDB_A001206PGDB_C032044PGDB_AS000657View
2D structure for PGDB_C032029
Dmax-=94.9%0.02 nM-VAV1--WO2026119120A1PGDB_A001360PGDB_C032029PGDB_AS000657View
2D structure for PGDB_C032060
Dmax-=95.6%0.02 nM-VAV1--WO2026119120A1PGDB_A001445PGDB_C032060PGDB_AS000657View
2D structure for PGDB_C032057
Dmax-=96%0.02 nM-VAV1--WO2026119120A1PGDB_A001587PGDB_C032057PGDB_AS000657View
2D structure for PGDB_C032070
Dmax-=96.6%0.02 nM-VAV1--WO2026119120A1PGDB_A001897PGDB_C032070PGDB_AS000657View
2D structure for PGDB_C032047
Dmax-=95.4%0.02 nM-VAV1--WO2026119120A1PGDB_A002025PGDB_C032047PGDB_AS000657View
2D structure for PGDB_C032058
Dmax-=96.2%0.02 nM-VAV1--WO2026119120A1PGDB_A002103PGDB_C032058PGDB_AS000657View
2D structure for PGDB_C032027
Dmax-=89%0.02 nM-VAV1--WO2026119120A1PGDB_A002164PGDB_C032027PGDB_AS000657View
2D structure for PGDB_C032032
Dmax-=87.8%0.02 nM-VAV1--WO2026119120A1PGDB_A002235PGDB_C032032PGDB_AS000657View
2D structure for PGDB_C032050
Dmax-=92.7%0.02 nM-VAV1--WO2026119120A1PGDB_A002434PGDB_C032050PGDB_AS000657View
2D structure for PGDB_C032073
Dmax-=95.2%0.02 nM-VAV1--WO2026119120A1PGDB_A002643PGDB_C032073PGDB_AS000657View
2D structure for PGDB_C032049
Dmax-=97.5%0.02 nM-VAV1--WO2026119120A1PGDB_A002833PGDB_C032049PGDB_AS000657View
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