Assay context summary

Assay context

33 activity records
Activity compounds and values

Activity records

33 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000492
IC50-=3.511nM-GSPT1-MV-4-11CN117917402APGDB_A007276PGDB_C000492PGDB_AS000703View
2D structure for PGDB_C000478
IC50-=1150nM-GSPT1-MV-4-11CN117917402APGDB_A009326PGDB_C000478PGDB_AS000703View
2D structure for PGDB_C000481
IC50->10000nM-GSPT1-MV-4-11CN117917402APGDB_A011392PGDB_C000481PGDB_AS000703View
2D structure for PGDB_C000477
IC50-=222.8nM-GSPT1-MV-4-11CN117917402APGDB_A013245PGDB_C000477PGDB_AS000703View
2D structure for PGDB_C000495
IC50-=18.25nM-GSPT1-MV-4-11CN117917402APGDB_A013358PGDB_C000495PGDB_AS000703View
2D structure for PGDB_C000496
IC50-=9.611nM-GSPT1-MV-4-11CN117917402APGDB_A013454PGDB_C000496PGDB_AS000703View
2D structure for PGDB_C000473
IC50-=120.3nM-GSPT1-MV-4-11CN117917402APGDB_A014965PGDB_C000473PGDB_AS000703View
2D structure for PGDB_C000491
IC50-=48.8nM-GSPT1-MV-4-11CN117917402APGDB_A016229PGDB_C000491PGDB_AS000703View
2D structure for PGDB_C000482
IC50->10000nM-GSPT1-MV-4-11CN117917402APGDB_A018390PGDB_C000482PGDB_AS000703View
2D structure for PGDB_C000501
IC50->10000nM-GSPT1-MV-4-11CN117917402APGDB_A020633PGDB_C000501PGDB_AS000703View
2D structure for PGDB_C000498
IC50-=42.05nM-GSPT1-MV-4-11CN117917402APGDB_A023212PGDB_C000498PGDB_AS000703View
2D structure for PGDB_C000494
IC50-=49.56nM-GSPT1-MV-4-11CN117917402APGDB_A026131PGDB_C000494PGDB_AS000703View
2D structure for PGDB_C000497
IC50-=3.188nM-GSPT1-MV-4-11CN117917402APGDB_A026199PGDB_C000497PGDB_AS000703View
2D structure for PGDB_C000489
IC50-=29.49nM-GSPT1-MV-4-11CN117917402APGDB_A031853PGDB_C000489PGDB_AS000703View
2D structure for PGDB_C000479
IC50->10000nM-GSPT1-MV-4-11CN117917402APGDB_A035709PGDB_C000479PGDB_AS000703View
2D structure for PGDB_C000476
IC50->10000nM-GSPT1-MV-4-11CN117917402APGDB_A035796PGDB_C000476PGDB_AS000703View
2D structure for PGDB_C000484
IC50-=23.7nM-GSPT1-MV-4-11CN117917402APGDB_A037056PGDB_C000484PGDB_AS000703View
2D structure for PGDB_C000488
IC50-=7.601nM-GSPT1-MV-4-11CN117917402APGDB_A039954PGDB_C000488PGDB_AS000703View
2D structure for PGDB_C000475
IC50-=1697nM-GSPT1-MV-4-11CN117917402APGDB_A040212PGDB_C000475PGDB_AS000703View
2D structure for PGDB_C000502
IC50-=37.68nM-GSPT1-MV-4-11CN117917402APGDB_A043536PGDB_C000502PGDB_AS000703View