Assay
PGDB_AS000716
System: cell_basedTarget: GSPT1Cell line: 293A
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | Dmax | - | = | 61 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A008466 | PGDB_C001077 | PGDB_AS000716 | View |
 | Dmax | - | = | 34 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A016927 | PGDB_C001078 | PGDB_AS000716 | View |
 | Dmax | - | = | 61 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A019445 | PGDB_C001070 | PGDB_AS000716 | View |
 | Dmax | - | = | 26 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A023175 | PGDB_C001076 | PGDB_AS000716 | View |
 | Dmax | - | = | 29 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A050997 | PGDB_C001073 | PGDB_AS000716 | View |
 | Dmax | - | = | 99.3 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A051270 | PGDB_C001072 | PGDB_AS000716 | View |
 | Dmax | - | = | 77 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A057259 | PGDB_C001074 | PGDB_AS000716 | View |
 | Dmax | - | = | 99.5 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A062242 | PGDB_C001075 | PGDB_AS000716 | View |
 | Dmax | - | = | 73 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A062585 | PGDB_C001079 | PGDB_AS000716 | View |
 | Dmax | - | = | 97.9 | % | Concentration series: 5000 nM, 1000 nM, 200 nM, 40 nM, 8 nM, 1.6 nM, 0.32 nM, 0.064 nM, 0.0128 nM, 0 nM | 6 h | GSPT1 | - | 293A | CN121591645A | PGDB_A068868 | PGDB_C001071 | PGDB_AS000716 | View |