Assay context summary

Assay context

58 activity records
Activity compounds and values

Activity records

58 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C024745
Dmax-=92%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000048PGDB_C024745PGDB_AS000765View
2D structure for PGDB_C024811
Dmax-=96.1%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000067PGDB_C024811PGDB_AS000765View
2D structure for PGDB_C024742
Dmax-=88.5%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000198PGDB_C024742PGDB_AS000765View
2D structure for PGDB_C024818
Dmax-=103.9%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000247PGDB_C024818PGDB_AS000765View
2D structure for PGDB_C024817
Dmax-=96.9%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000327PGDB_C024817PGDB_AS000765View
2D structure for PGDB_C030155
Dmax-=96.6%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000331PGDB_C030155PGDB_AS000765View
2D structure for PGDB_C024758
Dmax-=100%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A000486PGDB_C024758PGDB_AS000765View
2D structure for PGDB_C024762
Dmax-=97.8%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A001044PGDB_C024762PGDB_AS000765View
2D structure for PGDB_C010388
Dmax-=95.62%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A001431PGDB_C010388PGDB_AS000765View
2D structure for PGDB_C024757
Dmax-=104.4%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A002082PGDB_C024757PGDB_AS000765View
2D structure for PGDB_C024752
Dmax-=108.3%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A002300PGDB_C024752PGDB_AS000765View
2D structure for PGDB_C024802
Dmax-=100%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A002493PGDB_C024802PGDB_AS000765View
2D structure for PGDB_C024754
Dmax-=98.8%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A002837PGDB_C024754PGDB_AS000765View
2D structure for PGDB_C024764
Dmax-=91.2%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A002957PGDB_C024764PGDB_AS000765View
2D structure for PGDB_C024765
Dmax-=94.7%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003161PGDB_C024765PGDB_AS000765View
2D structure for PGDB_C024749
Dmax-=89.3%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003207PGDB_C024749PGDB_AS000765View
2D structure for PGDB_C024761
Dmax-=89.6%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003379PGDB_C024761PGDB_AS000765View
2D structure for PGDB_C024799
Dmax-=105.4%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003518PGDB_C024799PGDB_AS000765View
2D structure for PGDB_C024804
Dmax-=95.8%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003671PGDB_C024804PGDB_AS000765View
2D structure for PGDB_C024807
Dmax-=86.2%Concentration range: 1000 nM-VAV1-JurkatWO2026061428A1PGDB_A003719PGDB_C024807PGDB_AS000765View