Assay context summary

Assay context

600 activity records
Activity compounds and values

Activity records

600 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C004917
IC50-<10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007079PGDB_C004917PGDB_AS000952View
2D structure for PGDB_C005098
IC50-<10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007213PGDB_C005098PGDB_AS000952View
2D structure for PGDB_C005187
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007231PGDB_C005187PGDB_AS000952View
2D structure for PGDB_C004972
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007780PGDB_C004972PGDB_AS000952View
2D structure for PGDB_C005254
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007900PGDB_C005254PGDB_AS000952View
2D structure for PGDB_C005002
IC50-=10-100nM-GSPT1-MOLM-13WO2022073469A1PGDB_A007936PGDB_C005002PGDB_AS000952View
2D structure for PGDB_C004783
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A007959PGDB_C004783PGDB_AS000952View
2D structure for PGDB_C005222
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008031PGDB_C005222PGDB_AS000952View
2D structure for PGDB_C004856
IC50-=10-100nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008069PGDB_C004856PGDB_AS000952View
2D structure for PGDB_C004900
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A008143PGDB_C004900PGDB_AS000952View
2D structure for PGDB_C004884
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A008147PGDB_C004884PGDB_AS000952View
2D structure for PGDB_C005231
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A008151PGDB_C005231PGDB_AS000952View
2D structure for PGDB_C005263
IC50-<10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008197PGDB_C005263PGDB_AS000952View
2D structure for PGDB_C004719
IC50-<10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008340PGDB_C004719PGDB_AS000952View
2D structure for PGDB_C005009
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A008416PGDB_C005009PGDB_AS000952View
2D structure for PGDB_C004926
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008535PGDB_C004926PGDB_AS000952View
2D structure for PGDB_C004760
IC50->=1uM-GSPT1-MOLM-13WO2022073469A1PGDB_A008665PGDB_C004760PGDB_AS000952View
2D structure for PGDB_C004768
IC50-=100-1000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008686PGDB_C004768PGDB_AS000952View
2D structure for PGDB_C005280
IC50-=10-100nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008713PGDB_C005280PGDB_AS000952View
2D structure for PGDB_C005094
IC50-<10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008844PGDB_C005094PGDB_AS000952View