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Cc1nn([C@H]2C[C@@H](CCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1-c1cnc2cc(N3CCN(C)CC3)ccc2n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A007079 | PGDB_C004917 | PGDB_AS000952 | View | |
| IC50 | - | = | 10-100 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A009684 | PGDB_C004917 | PGDB_AS000609 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A074884 | PGDB_C004917 | PGDB_AS000571 | View | |
| IC50 | - | < | 10 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A077613 | PGDB_C004917 | PGDB_AS002199 | View |