Assay
PGDB_AS000953
System: cell_basedCell line: Hep3B2.7-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 500-1000 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A020153 | PGDB_C025964 | PGDB_AS000953 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A035721 | PGDB_C025966 | PGDB_AS000953 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A055085 | PGDB_C025963 | PGDB_AS000953 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A055724 | PGDB_C025962 | PGDB_AS000953 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A064220 | PGDB_C025965 | PGDB_AS000953 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Hep3B2.7-1 | CN116239566A | PGDB_A074870 | PGDB_C025961 | PGDB_AS000953 | View |