Assay

PGDB_AS000988

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

22 activity records
Assay familybinding
Systembiochemical
ReadoutKd
TargetCRBN | DDB1
E3CRBN | DDB1
OrganismHomo sapiens
Technologyfluorescence
Activity compounds and values

Activity records

22 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007393
Kd-=0.023uM-—CRBNCRBN-EP3556760A1PGDB_A009560PGDB_C007393PGDB_AS000988View
2D structure for PGDB_C007385
Kd-=0.017uM-—CRBNCRBN-EP3556760A1PGDB_A012816PGDB_C007385PGDB_AS000988View
2D structure for PGDB_C007383
Kd-=0.002uM-—CRBNCRBN-EP3556760A1PGDB_A013644PGDB_C007383PGDB_AS000988View
2D structure for PGDB_C007403
Kd-=0.006uM-—CRBNCRBN-EP3556760A1PGDB_A016107PGDB_C007403PGDB_AS000988View
2D structure for PGDB_C007404
Kd-=0.006uM-—CRBNCRBN-EP3556760A1PGDB_A017791PGDB_C007404PGDB_AS000988View
2D structure for PGDB_C007384
Kd-=0.002uM-—CRBNCRBN-EP3556760A1PGDB_A020924PGDB_C007384PGDB_AS000988View
2D structure for PGDB_C025999
Kd-=0.007uM-—CRBNCRBN-EP3556760A1PGDB_A024556PGDB_C025999PGDB_AS000988View
2D structure for PGDB_C026003
Kd-<0.001uM-—CRBNCRBN-EP3556760A1PGDB_A030028PGDB_C026003PGDB_AS000988View
2D structure for PGDB_C007389
Kd-=0.001uM-—CRBNCRBN-EP3556760A1PGDB_A032428PGDB_C007389PGDB_AS000988View
2D structure for PGDB_C026001
Kd-=0.002uM-—CRBNCRBN-EP3556760A1PGDB_A036296PGDB_C026001PGDB_AS000988View
2D structure for PGDB_C007391
Kd-=0.016uM-—CRBNCRBN-EP3556760A1PGDB_A042542PGDB_C007391PGDB_AS000988View
2D structure for PGDB_C007388
Kd-=0.021uM-—CRBNCRBN-EP3556760A1PGDB_A042760PGDB_C007388PGDB_AS000988View
2D structure for PGDB_C007396
Kd-=0.006uM-—CRBNCRBN-EP3556760A1PGDB_A043155PGDB_C007396PGDB_AS000988View
2D structure for PGDB_C007402
Kd-=0.028uM-—CRBNCRBN-EP3556760A1PGDB_A047173PGDB_C007402PGDB_AS000988View
2D structure for PGDB_C007399
Kd-=0.015uM-—CRBNCRBN-EP3556760A1PGDB_A048840PGDB_C007399PGDB_AS000988View
2D structure for PGDB_C007387
Kd-=0.027uM-—CRBNCRBN-EP3556760A1PGDB_A057013PGDB_C007387PGDB_AS000988View
2D structure for PGDB_C007400
Kd-=0.006uM-—CRBNCRBN-EP3556760A1PGDB_A066296PGDB_C007400PGDB_AS000988View
2D structure for PGDB_C007390
Kd-<0.001uM-—CRBNCRBN-EP3556760A1PGDB_A066768PGDB_C007390PGDB_AS000988View
2D structure for PGDB_C007386
Kd-=0.034uM-—CRBNCRBN-EP3556760A1PGDB_A068908PGDB_C007386PGDB_AS000988View
2D structure for PGDB_C011112
Kd-=0.011uM-—CRBNCRBN-EP3556760A1PGDB_A071403PGDB_C011112PGDB_AS000988View
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