Assay

PGDB_AS001033

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

267 activity records
Assay familybiochemical
Systembiochemical
ReadoutEC50
TargetCRBN | DDB1
E3CRBN | DDB1
TechnologyHTRF
Activity compounds and values

Activity records

267 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020302
EC50-=0.09uM-—CRBNCRBN-WO2025024521A1PGDB_A007237PGDB_C020302PGDB_AS001033View
2D structure for PGDB_C020440
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A007581PGDB_C020440PGDB_AS001033View
2D structure for PGDB_C020382
EC50-=0.09uM-—CRBNCRBN-WO2025024521A1PGDB_A008063PGDB_C020382PGDB_AS001033View
2D structure for PGDB_C020357
EC50-=0.18uM-—CRBNCRBN-WO2025024521A1PGDB_A008266PGDB_C020357PGDB_AS001033View
2D structure for PGDB_C020452
EC50-=0.24uM-—CRBNCRBN-WO2025024521A1PGDB_A008558PGDB_C020452PGDB_AS001033View
2D structure for PGDB_C020429
EC50-=0.08uM-—CRBNCRBN-WO2025024521A1PGDB_A009164PGDB_C020429PGDB_AS001033View
2D structure for PGDB_C020324
EC50-=0.17uM-—CRBNCRBN-WO2025024521A1PGDB_A009191PGDB_C020324PGDB_AS001033View
2D structure for PGDB_C020317
EC50-=0.14uM-—CRBNCRBN-WO2025024521A1PGDB_A009437PGDB_C020317PGDB_AS001033View
2D structure for PGDB_C020444
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A009652PGDB_C020444PGDB_AS001033View
2D structure for PGDB_C020294
EC50-=0.29uM-—CRBNCRBN-WO2025024521A1PGDB_A009665PGDB_C020294PGDB_AS001033View
2D structure for PGDB_C020454
EC50-=0.26uM-—CRBNCRBN-WO2025024521A1PGDB_A010206PGDB_C020454PGDB_AS001033View
2D structure for PGDB_C020336
EC50-=0.25uM-—CRBNCRBN-WO2025024521A1PGDB_A010470PGDB_C020336PGDB_AS001033View
2D structure for PGDB_C020404
EC50-=0.14uM-—CRBNCRBN-WO2025024521A1PGDB_A010596PGDB_C020404PGDB_AS001033View
2D structure for PGDB_C020422
EC50-=0.07uM-—CRBNCRBN-WO2025024521A1PGDB_A010725PGDB_C020422PGDB_AS001033View
2D structure for PGDB_C020360
EC50-=0.1uM-—CRBNCRBN-WO2025024521A1PGDB_A011168PGDB_C020360PGDB_AS001033View
2D structure for PGDB_C020400
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A012318PGDB_C020400PGDB_AS001033View
2D structure for PGDB_C020303
EC50-=0.04uM-—CRBNCRBN-WO2025024521A1PGDB_A012543PGDB_C020303PGDB_AS001033View
2D structure for PGDB_C020433
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A012572PGDB_C020433PGDB_AS001033View
2D structure for PGDB_C020439
EC50-=0.12uM-—CRBNCRBN-WO2025024521A1PGDB_A012954PGDB_C020439PGDB_AS001033View
2D structure for PGDB_C020392
EC50-=0.08uM-—CRBNCRBN-WO2025024521A1PGDB_A012956PGDB_C020392PGDB_AS001033View
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