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SIMM · NJU
Assay
PGDB_AS001169
System: cell_based
Target: IKZF2
Cell line: 293GT
Assay context summary
Assay context
143 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF2
E3
CRBN
Cell line
293GT
Organism
Homo sapiens
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
143 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
1.08
uM
-
—
-
-
293GT
CN111051298A
PGDB_A007428
PGDB_C022729
PGDB_AS001169
View
EC50
-
=
0.031
uM
-
—
-
-
293GT
CN111051298A
PGDB_A008080
PGDB_C022761
PGDB_AS001169
View
EC50
-
=
0.11
uM
-
—
-
-
293GT
CN111051298A
PGDB_A008607
PGDB_C022714
PGDB_AS001169
View
EC50
-
=
0.17
uM
-
—
-
-
293GT
CN111051298A
PGDB_A008963
PGDB_C022735
PGDB_AS001169
View
EC50
-
=
0.24
uM
-
—
-
-
293GT
CN111051298A
PGDB_A011233
PGDB_C022748
PGDB_AS001169
View
EC50
-
=
0.013
uM
-
—
-
-
293GT
CN111051298A
PGDB_A012236
PGDB_C022670
PGDB_AS001169
View
EC50
-
=
0.067
uM
-
—
-
-
293GT
CN111051298A
PGDB_A012483
PGDB_C022705
PGDB_AS001169
View
EC50
-
=
0.017
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013055
PGDB_C022662
PGDB_AS001169
View
EC50
-
=
0.006
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013162
PGDB_C022640
PGDB_AS001169
View
EC50
-
=
0.05
uM
-
—
-
-
293GT
CN111051298A
PGDB_A013740
PGDB_C022754
PGDB_AS001169
View
EC50
-
=
0.21
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014041
PGDB_C022677
PGDB_AS001169
View
EC50
-
=
0.039
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014210
PGDB_C022690
PGDB_AS001169
View
EC50
-
=
9.8
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014377
PGDB_C022725
PGDB_AS001169
View
EC50
-
=
0.036
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014492
PGDB_C022712
PGDB_AS001169
View
EC50
-
=
0.012
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014606
PGDB_C022653
PGDB_AS001169
View
EC50
-
=
0.03
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014689
PGDB_C022674
PGDB_AS001169
View
EC50
-
=
0.013
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014775
PGDB_C022633
PGDB_AS001169
View
EC50
-
=
0.029
uM
-
—
-
-
293GT
CN111051298A
PGDB_A014885
PGDB_C022747
PGDB_AS001169
View
EC50
-
=
0.005
uM
-
—
-
-
293GT
CN111051298A
PGDB_A015198
PGDB_C022685
PGDB_AS001169
View
EC50
-
=
0.018
uM
-
—
-
-
293GT
CN111051298A
PGDB_A015292
PGDB_C022652
PGDB_AS001169
View