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O=C1CCC(N2Cc3cc(C4CCN(Cc5ccc(C(F)F)cc5)CC4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.012 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A014606 | PGDB_C022653 | PGDB_AS001169 | View | |
| % Degradation | - | = | 75.0 | % | 10 uM | 24 h | - | - | 293GT | CN111051298A | PGDB_A018012 | PGDB_C022653 | PGDB_AS002112 | View | |
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A020551 | PGDB_C022653 | PGDB_AS000334 | View | |
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A026723 | PGDB_C022653 | PGDB_AS002316 | View |