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SIMM · NJU
Assay
PGDB_AS001249
System: cell_based
Target: CCNK
Cell line: HEK293T_Nluc_CCNK-tagged
Assay context summary
Assay context
51 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
CCNK
E3
Not specified
Cell line
HEK293T_Nluc_CCNK-tagged
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
51 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A010593
PGDB_C010853
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A012115
PGDB_C010858
PGDB_AS001249
View
DC50
-
<
10
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A013253
PGDB_C010872
PGDB_AS001249
View
DC50
-
=
1-100
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A015420
PGDB_C010889
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A015677
PGDB_C010862
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A015770
PGDB_C010885
PGDB_AS001249
View
DC50
-
=
1-100
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A021595
PGDB_C010867
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A022708
PGDB_C010861
PGDB_AS001249
View
DC50
-
=
1-100
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A022766
PGDB_C010855
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A025443
PGDB_C010890
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A027148
PGDB_C010866
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A027393
PGDB_C010863
PGDB_AS001249
View
DC50
-
<
10
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A028214
PGDB_C010875
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A028920
PGDB_C010846
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A031288
PGDB_C010869
PGDB_AS001249
View
DC50
-
=
0.1-1
uM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A031524
PGDB_C010856
PGDB_AS001249
View
DC50
-
<
10
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A031942
PGDB_C010874
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A032738
PGDB_C010893
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A033574
PGDB_C010894
PGDB_AS001249
View
DC50
-
=
10-100
nM
-
—
CCNK
-
HEK293T_Nluc_CCNK-tagged
WO2025104236
PGDB_A033856
PGDB_C010888
PGDB_AS001249
View