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SIMM · NJU
Assay
PGDB_AS001390
System: cell_based
Target: VAV1
Cell line: Jurkat
Assay context summary
Assay context
61 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Cell line
Jurkat
Organism
Homo sapiens
Technology
fluorescence
Activity compounds and values
Activity records
61 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A000236
PGDB_C030185
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A000482
PGDB_C024824
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A000692
PGDB_C024762
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A000926
PGDB_C024741
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001038
PGDB_C024754
PGDB_AS001390
View
DC50
-
=
50-500
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001346
PGDB_C024752
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001451
PGDB_C024760
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001485
PGDB_C024815
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001531
PGDB_C024805
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001591
PGDB_C024822
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001688
PGDB_C024745
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A001694
PGDB_C025999
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A002011
PGDB_C024799
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A002511
PGDB_C024739
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A002534
PGDB_C030186
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A002763
PGDB_C026003
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A002871
PGDB_C024796
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A003047
PGDB_C024814
PGDB_AS001390
View
DC50
-
=
50-500
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A003261
PGDB_C024764
PGDB_AS001390
View
DC50
-
<=
50
nM
-
—
VAV1
-
Jurkat
WO2026061428A1
PGDB_A003399
PGDB_C024744
PGDB_AS001390
View