Assay

PGDB_AS001469

System: biochemicalTarget: CRBN
Assay context summary

Assay context

19 activity records
Assay familybiochemical
Systembiochemical
ReadoutEC50
TargetCRBN
E3CRBN
TechnologyHTRF
Activity compounds and values

Activity records

19 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020449
EC50-=0.19uM-—CRBNCRBN-WO2025024521A1PGDB_A012203PGDB_C020449PGDB_AS001469View
2D structure for PGDB_C020451
EC50-=0.19uM-—CRBNCRBN-WO2025024521A1PGDB_A015534PGDB_C020451PGDB_AS001469View
2D structure for PGDB_C020439
EC50-=0.12uM-—CRBNCRBN-WO2025024521A1PGDB_A016195PGDB_C020439PGDB_AS001469View
2D structure for PGDB_C020446
EC50-=0.25uM-—CRBNCRBN-WO2025024521A1PGDB_A023667PGDB_C020446PGDB_AS001469View
2D structure for PGDB_C020453
EC50-=0.29uM-—CRBNCRBN-WO2025024521A1PGDB_A033676PGDB_C020453PGDB_AS001469View
2D structure for PGDB_C020440
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A037659PGDB_C020440PGDB_AS001469View
2D structure for PGDB_C020447
EC50-=10uM-—CRBNCRBN-WO2025024521A1PGDB_A039643PGDB_C020447PGDB_AS001469View
2D structure for PGDB_C020438
EC50-=0.12uM-—CRBNCRBN-WO2025024521A1PGDB_A043121PGDB_C020438PGDB_AS001469View
2D structure for PGDB_C020442
EC50-=0.1uM-—CRBNCRBN-WO2025024521A1PGDB_A044179PGDB_C020442PGDB_AS001469View
2D structure for PGDB_C020455
EC50-=0.11uM-—CRBNCRBN-WO2025024521A1PGDB_A053644PGDB_C020455PGDB_AS001469View
2D structure for PGDB_C020445
EC50-=0.23uM-—CRBNCRBN-WO2025024521A1PGDB_A060447PGDB_C020445PGDB_AS001469View
2D structure for PGDB_C020450
EC50-=0.18uM-—CRBNCRBN-WO2025024521A1PGDB_A065122PGDB_C020450PGDB_AS001469View
2D structure for PGDB_C020444
EC50-=0.52uM-—CRBNCRBN-WO2025024521A1PGDB_A069516PGDB_C020444PGDB_AS001469View
2D structure for PGDB_C020435
EC50-=0.08uM-—CRBNCRBN-WO2025024521A1PGDB_A070214PGDB_C020435PGDB_AS001469View
2D structure for PGDB_C020452
EC50-=0.35uM-—CRBNCRBN-WO2025024521A1PGDB_A070251PGDB_C020452PGDB_AS001469View
2D structure for PGDB_C020448
EC50-=0.21uM-—CRBNCRBN-WO2025024521A1PGDB_A072449PGDB_C020448PGDB_AS001469View
2D structure for PGDB_C020437
EC50-=0.13uM-—CRBNCRBN-WO2025024521A1PGDB_A076120PGDB_C020437PGDB_AS001469View
2D structure for PGDB_C020454
EC50-=0.26uM-—CRBNCRBN-WO2025024521A1PGDB_A076975PGDB_C020454PGDB_AS001469View
2D structure for PGDB_C020436
EC50-=0.1uM-—CRBNCRBN-WO2025024521A1PGDB_A077568PGDB_C020436PGDB_AS001469View
Page 1 of 1 · 19 records