Assay
PGDB_AS001477
System: cell_basedCell line: BT-474
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A011867 | PGDB_C001024 | PGDB_AS001477 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A027931 | PGDB_C001019 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A036830 | PGDB_C001022 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A043615 | PGDB_C001018 | PGDB_AS001477 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A050080 | PGDB_C001025 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A053304 | PGDB_C001021 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A060537 | PGDB_C001020 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A062808 | PGDB_C001023 | PGDB_AS001477 | View | |
| IC50 | - | = | 10-30 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A066198 | PGDB_C001026 | PGDB_AS001477 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | BT-474 | CN121219280A | PGDB_A070486 | PGDB_C001027 | PGDB_AS001477 | View |