Assay
PGDB_AS001576
System: cell_basedCell line: MDA-MB-231
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A021253 | PGDB_C025942 | PGDB_AS001576 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A021617 | PGDB_C025937 | PGDB_AS001576 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A023857 | PGDB_C025939 | PGDB_AS001576 | View | |
| IC50 | - | = | 50-100 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A036990 | PGDB_C025940 | PGDB_AS001576 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A037134 | PGDB_C025943 | PGDB_AS001576 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A051791 | PGDB_C025944 | PGDB_AS001576 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A056030 | PGDB_C025935 | PGDB_AS001576 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A068685 | PGDB_C025936 | PGDB_AS001576 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A075282 | PGDB_C025938 | PGDB_AS001576 | View |