Loading compound
Loading detail record from the SQLite release...
Loading detail record from the SQLite release...
CNC(=O)c1ccccc1Nc1cc(Nc2ccc(N3CCC(N4CCN(Cc5ccc6c(c5F)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2OC)ncc1C(F)(F)F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SR | CN116239566A | PGDB_A012602 | PGDB_C025936 | PGDB_AS001780 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A024946 | PGDB_C025936 | PGDB_AS001781 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | PC-9 | CN116239566A | PGDB_A031089 | PGDB_C025936 | PGDB_AS001387 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A054732 | PGDB_C025936 | PGDB_AS000686 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | MDA-MB-231 | CN116239566A | PGDB_A068685 | PGDB_C025936 | PGDB_AS001576 | View |