Assay

PGDB_AS001592

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

42 activity records
Assay familybinding
Systembiochemical
ReadoutKi
TargetCRBN | DDB1
E3CRBN | DDB1
Technologyfluorescence
Activity compounds and values

Activity records

42 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000078
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A007045PGDB_C000078PGDB_AS001592View
2D structure for PGDB_C000052
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A008863PGDB_C000052PGDB_AS001592View
2D structure for PGDB_C000079
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A011906PGDB_C000079PGDB_AS001592View
2D structure for PGDB_C000100
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A015704PGDB_C000100PGDB_AS001592View
2D structure for PGDB_C000097
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A018049PGDB_C000097PGDB_AS001592View
2D structure for PGDB_C000091
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A018606PGDB_C000091PGDB_AS001592View
2D structure for PGDB_C000064
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A019412PGDB_C000064PGDB_AS001592View
2D structure for PGDB_C000062
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A021525PGDB_C000062PGDB_AS001592View
2D structure for PGDB_C000096
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A026324PGDB_C000096PGDB_AS001592View
2D structure for PGDB_C000098
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A026325PGDB_C000098PGDB_AS001592View
2D structure for PGDB_C000075
Ki-=0.5-1uM-—CRBNCRBN-CN116457344APGDB_A026761PGDB_C000075PGDB_AS001592View
2D structure for PGDB_C000076
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A027946PGDB_C000076PGDB_AS001592View
2D structure for PGDB_C000085
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A031235PGDB_C000085PGDB_AS001592View
2D structure for PGDB_C000077
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A032933PGDB_C000077PGDB_AS001592View
2D structure for PGDB_C000065
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A034394PGDB_C000065PGDB_AS001592View
2D structure for PGDB_C000092
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A037225PGDB_C000092PGDB_AS001592View
2D structure for PGDB_C000053
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A040038PGDB_C000053PGDB_AS001592View
2D structure for PGDB_C000066
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A040386PGDB_C000066PGDB_AS001592View
2D structure for PGDB_C000089
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A041220PGDB_C000089PGDB_AS001592View
2D structure for PGDB_C000094
Ki-<0.5uM-—CRBNCRBN-CN116457344APGDB_A043754PGDB_C000094PGDB_AS001592View
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