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N[C@@H](Cc1cnc[nH]1)C(=O)NCc1ccc2c(c1)CN([C@H]1CCC(=O)NC1=O)C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ki | - | < | 0.5 | uM | - | — | CRBN | CRBN | - | CN116457344A | PGDB_A021525 | PGDB_C000062 | PGDB_AS001592 | View | |
| IC50 | - | > | 50 | uM | - | — | - | - | H929 | CN116457344A | PGDB_A027107 | PGDB_C000062 | PGDB_AS000797 | View | |
| IC50 | - | = | 0.1-1 | uM | - | — | - | - | Hep3B | CN116457344A | PGDB_A030293 | PGDB_C000062 | PGDB_AS001471 | View | |
| IC50 | - | = | 100-1000 | nM | - | — | - | - | Kelly | CN116457344A | PGDB_A042516 | PGDB_C000062 | PGDB_AS002343 | View | |
| IC50 | - | = | 0.1-1 | uM | - | — | - | - | KG-1 | CN116457344A | PGDB_A061261 | PGDB_C000062 | PGDB_AS000548 | View |