Assay
PGDB_AS001594
System: cell_basedTarget: ESR1Cell line: MCF-7
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.36 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A008610 | PGDB_C006617 | PGDB_AS001594 | View | |
| IC50 | - | = | 0.18 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A021093 | PGDB_C006618 | PGDB_AS001594 | View | |
| IC50 | - | = | 0.89 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A022645 | PGDB_C006613 | PGDB_AS001594 | View | |
| IC50 | - | = | 0.69 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A030883 | PGDB_C006614 | PGDB_AS001594 | View | |
| IC50 | - | = | 1.5 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A038756 | PGDB_C006619 | PGDB_AS001594 | View | |
| IC50 | - | = | 1 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A051669 | PGDB_C006616 | PGDB_AS001594 | View | |
| IC50 | - | = | 0.32 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A066766 | PGDB_C006620 | PGDB_AS001594 | View | |
| IC50 | - | = | 1.1 | nM | - | — | ESR1 | - | MCF-7 | CN115260206A | PGDB_A068762 | PGDB_C006615 | PGDB_AS001594 | View |