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SIMM · NJU
Assay
PGDB_AS001673
System: cell_based
Cell line: Jurkat
Assay context summary
Assay context
124 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
E3
Not specified
Cell line
Jurkat
Organism
Homo sapiens
Detection target
protein_degradation
Activity compounds and values
Activity records
124 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A000630
PGDB_C031718
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001077
PGDB_C031823
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001230
PGDB_C031815
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001285
PGDB_C031791
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001710
PGDB_C031831
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001838
PGDB_C031700
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001848
PGDB_C031829
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001885
PGDB_C031732
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A001957
PGDB_C031807
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002007
PGDB_C031851
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002311
PGDB_C031812
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002371
PGDB_C031689
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002452
PGDB_C031709
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002520
PGDB_C031730
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002630
PGDB_C031723
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002844
PGDB_C031813
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002874
PGDB_C031827
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002876
PGDB_C031802
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002881
PGDB_C031838
PGDB_AS001673
View
% Degradation
-
>
50
%
10 nM
-
VAV1
-
Jurkat
WO2026114367A1
PGDB_A002941
PGDB_C031843
PGDB_AS001673
View