Assay context summary

Assay context

124 activity records
Activity compounds and values

Activity records

124 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031718
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A000630PGDB_C031718PGDB_AS001673View
2D structure for PGDB_C031823
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001077PGDB_C031823PGDB_AS001673View
2D structure for PGDB_C031815
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001230PGDB_C031815PGDB_AS001673View
2D structure for PGDB_C031791
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001285PGDB_C031791PGDB_AS001673View
2D structure for PGDB_C031831
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001710PGDB_C031831PGDB_AS001673View
2D structure for PGDB_C031700
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001838PGDB_C031700PGDB_AS001673View
2D structure for PGDB_C031829
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001848PGDB_C031829PGDB_AS001673View
2D structure for PGDB_C031732
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001885PGDB_C031732PGDB_AS001673View
2D structure for PGDB_C031807
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A001957PGDB_C031807PGDB_AS001673View
2D structure for PGDB_C031851
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002007PGDB_C031851PGDB_AS001673View
2D structure for PGDB_C031812
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002311PGDB_C031812PGDB_AS001673View
2D structure for PGDB_C031689
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002371PGDB_C031689PGDB_AS001673View
2D structure for PGDB_C031709
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002452PGDB_C031709PGDB_AS001673View
2D structure for PGDB_C031730
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002520PGDB_C031730PGDB_AS001673View
2D structure for PGDB_C031723
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002630PGDB_C031723PGDB_AS001673View
2D structure for PGDB_C031813
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002844PGDB_C031813PGDB_AS001673View
2D structure for PGDB_C031827
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002874PGDB_C031827PGDB_AS001673View
2D structure for PGDB_C031802
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002876PGDB_C031802PGDB_AS001673View
2D structure for PGDB_C031838
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002881PGDB_C031838PGDB_AS001673View
2D structure for PGDB_C031843
% Degradation->50%10 nM-VAV1-JurkatWO2026114367A1PGDB_A002941PGDB_C031843PGDB_AS001673View