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SIMM · NJU
Assay
PGDB_AS001708
System: cell_based
Assay context summary
Assay context
36 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Detection target
protein_degradation
Activity compounds and values
Activity records
36 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
0.12
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A008862
PGDB_C025580
PGDB_AS001708
View
Dmax
-
=
0.1
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A012732
PGDB_C025596
PGDB_AS001708
View
Dmax
-
=
0.28
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A012947
PGDB_C025587
PGDB_AS001708
View
Dmax
-
=
0.44
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A013015
PGDB_C025583
PGDB_AS001708
View
Dmax
-
=
0.12
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A018748
PGDB_C025567
PGDB_AS001708
View
Dmax
-
=
0.24
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A022202
PGDB_C025574
PGDB_AS001708
View
Dmax
-
=
0.43
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A023091
PGDB_C025570
PGDB_AS001708
View
Dmax
-
=
0.13
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A023449
PGDB_C025571
PGDB_AS001708
View
Dmax
-
=
0.03
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A026401
PGDB_C025595
PGDB_AS001708
View
Dmax
-
=
0.07
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A030170
PGDB_C025577
PGDB_AS001708
View
Dmax
-
=
0.1
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A030351
PGDB_C025565
PGDB_AS001708
View
Dmax
-
=
0.04
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A032924
PGDB_C025576
PGDB_AS001708
View
Dmax
-
=
0.34
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A032976
PGDB_C025572
PGDB_AS001708
View
Dmax
-
=
0.09
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A033681
PGDB_C025588
PGDB_AS001708
View
Dmax
-
=
0.54
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A035376
PGDB_C025566
PGDB_AS001708
View
Dmax
-
=
0.21
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A038109
PGDB_C025575
PGDB_AS001708
View
Dmax
-
=
0.18
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A038504
PGDB_C025593
PGDB_AS001708
View
Dmax
-
=
0.18
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A039699
PGDB_C009602
PGDB_AS001708
View
Dmax
-
=
0.18
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A042692
PGDB_C025569
PGDB_AS001708
View
Dmax
-
=
0.09
%
-
-
-
CRBN
-
EP4683934A1
PGDB_A045506
PGDB_C009602
PGDB_AS001708
View