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O=C1CCC(N2C(=O)c3ccc(O)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.114 | uM | - | — | PARG | - | - | WO2026062066A1 | PGDB_A000487 | PGDB_C025567 | PGDB_AS002282 | View | |
| EC50 | - | > | 20 | uM | - | — | PARG | - | NCIH-460 | WO2026062066A1 | PGDB_A004835 | PGDB_C025567 | PGDB_AS002426 | View | |
| DC50 | - | = | 26.91534803926914 | nM | - | — | - | - | - | EP4683934A1 | PGDB_A011982 | PGDB_C025567 | PGDB_AS000564 | View | |
| Dmax | - | = | 0.12 | % | - | - | - | CRBN | - | EP4683934A1 | PGDB_A018748 | PGDB_C025567 | PGDB_AS001708 | View | |
| DC50 | - | = | 20.892961308540407 | nM | - | — | - | - | - | EP4683934A1 | PGDB_A025391 | PGDB_C025567 | PGDB_AS002010 | View | |
| IC50 | - | = | 40.7380277804113 | nM | - | — | - | - | - | EP4683934A1 | PGDB_A065523 | PGDB_C025567 | PGDB_AS002416 | View | |
| EC50 | - | > | 20 | uM | - | — | PARG | - | U2OS | WO2026062066A1 | PGDB_A081137 | PGDB_C025567 | PGDB_AS002468 | View |