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SIMM · NJU
Assay
PGDB_AS001734
System: cell_based
Target: GSPT1
Cell line: 293GT
Assay context summary
Assay context
43 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
GSPT1
E3
Not specified
Cell line
293GT
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
43 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A007417
PGDB_C008909
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A011363
PGDB_C008798
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A013972
PGDB_C008884
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A014753
PGDB_C008708
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A016970
PGDB_C008756
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A017606
PGDB_C008775
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A021915
PGDB_C008767
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A024071
PGDB_C008857
PGDB_AS001734
View
EC50
-
>
50
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A026407
PGDB_C008769
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A026980
PGDB_C008766
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A033787
PGDB_C008902
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A034529
PGDB_C008802
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A039452
PGDB_C008861
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A039767
PGDB_C008907
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A041566
PGDB_C008762
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A044040
PGDB_C008778
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A044444
PGDB_C008755
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A044511
PGDB_C008917
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A045636
PGDB_C008840
PGDB_AS001734
View
EC50
-
>
30
mM
-
—
GSPT1
-
293GT
KR20210031680A
PGDB_A046754
PGDB_C008924
PGDB_AS001734
View