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Compound
PGDB_C008708
8 activity records2 related patents
2D structure
O=C1CCC(N2Cc3cc(O[C@H]4CCCC[C@@H]4NCc4ccccc4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 30 | mM | - | — | GSPT1 | - | 293GT | KR20210031680A | PGDB_A014753 | PGDB_C008708 | PGDB_AS001734 | View |
| EC50 | - | = | 0.016 | mM | - | — | IKZF2 | - | 293GT | KR20210031680A | PGDB_A022407 | PGDB_C008708 | PGDB_AS001244 | View |
| % Degradation | - | = | 80 | % | 10 uM | 24 h | IKZF2 | - | 293GT | KR20210031680A | PGDB_A033873 | PGDB_C008708 | PGDB_AS000887 | View |
| % Degradation | - | = | 0.2 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A048710 | PGDB_C008708 | PGDB_AS000906 | View |
| EC50 | - | > | 50 | mM | - | — | IKZF1 | - | 293GT | KR20210031680A | PGDB_A051683 | PGDB_C008708 | PGDB_AS002284 | View |
| EC50 | - | = | 0.057 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A059326 | PGDB_C008708 | PGDB_AS001535 | View |
| EC50 | - | > | 50 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A060627 | PGDB_C008708 | PGDB_AS002086 | View |
| Dmax | - | = | 84 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A065077 | PGDB_C008708 | PGDB_AS000211 | View |