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SIMM · NJU
Assay
PGDB_AS001788
System: cell_based
Target: IKZF1
Cell line: HEK293
Assay context summary
Assay context
158 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF1
E3
Not specified
Cell line
HEK293
Detection target
protein_degradation
Activity compounds and values
Activity records
158 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.246
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A007928
PGDB_C005924
PGDB_AS001788
View
EC50
-
=
0.121
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008108
PGDB_C006007
PGDB_AS001788
View
EC50
-
=
0.07
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008215
PGDB_C005952
PGDB_AS001788
View
EC50
-
=
0.053
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008818
PGDB_C005875
PGDB_AS001788
View
EC50
-
=
0.023
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A008884
PGDB_C005881
PGDB_AS001788
View
EC50
-
=
0.07
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009078
PGDB_C005934
PGDB_AS001788
View
EC50
-
=
0.005
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009136
PGDB_C006012
PGDB_AS001788
View
EC50
-
=
0.038
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009210
PGDB_C005911
PGDB_AS001788
View
EC50
-
=
0.146
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009214
PGDB_C005998
PGDB_AS001788
View
EC50
-
=
0.047
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009711
PGDB_C005917
PGDB_AS001788
View
EC50
-
=
0.048
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A009861
PGDB_C005996
PGDB_AS001788
View
EC50
-
=
0.054
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A010279
PGDB_C005899
PGDB_AS001788
View
EC50
-
=
0.164
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A010393
PGDB_C005968
PGDB_AS001788
View
EC50
-
=
0.026
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A010691
PGDB_C005974
PGDB_AS001788
View
EC50
-
=
0.003
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A010812
PGDB_C005969
PGDB_AS001788
View
EC50
-
=
0.003
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A011568
PGDB_C006003
PGDB_AS001788
View
EC50
-
=
0.107
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A011654
PGDB_C005967
PGDB_AS001788
View
EC50
-
=
0.289
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A011832
PGDB_C005920
PGDB_AS001788
View
EC50
-
=
0.027
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A012046
PGDB_C006004
PGDB_AS001788
View
EC50
-
=
0.058
uM
-
—
IKZF1
-
HEK293
AU2022419982A1
PGDB_A013497
PGDB_C006022
PGDB_AS001788
View