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Compound
PGDB_C005996
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(CN[C@@H]4CCCN(Cc5ccccn5)C4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.048 | uM | - | — | IKZF1 | - | HEK293 | AU2022419982A1 | PGDB_A009861 | PGDB_C005996 | PGDB_AS001788 | View |
| EC50 | - | = | 0.138 | uM | - | — | IKZF2 | - | HEK293 | AU2022419982A1 | PGDB_A009898 | PGDB_C005996 | PGDB_AS002057 | View |
| Dmax | - | = | 97 | % | - | 24 h | IKZF1 | - | HEK293 | AU2022419982A1 | PGDB_A028002 | PGDB_C005996 | PGDB_AS000645 | View |
| Dmax | - | = | 97 | % | - | 24 h | IKZF2 | - | HEK293 | AU2022419982A1 | PGDB_A072235 | PGDB_C005996 | PGDB_AS000473 | View |