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SIMM · NJU
Assay
PGDB_AS001980
System: cell_based
Target: KRAS
Assay context summary
Assay context
57 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
KRAS
E3
Not specified
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
57 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
79
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000212
PGDB_C031966
PGDB_AS001980
View
Dmax
-
=
66
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000408
PGDB_C031989
PGDB_AS001980
View
Dmax
-
=
77
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000696
PGDB_C031963
PGDB_AS001980
View
Dmax
-
=
84
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000724
PGDB_C031941
PGDB_AS001980
View
Dmax
-
=
80
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000813
PGDB_C031970
PGDB_AS001980
View
Dmax
-
=
65
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000922
PGDB_C031960
PGDB_AS001980
View
Dmax
-
=
84
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000966
PGDB_C031949
PGDB_AS001980
View
Dmax
-
=
85
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001047
PGDB_C031955
PGDB_AS001980
View
Dmax
-
=
81
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001394
PGDB_C031972
PGDB_AS001980
View
Dmax
-
=
91
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001656
PGDB_C031996
PGDB_AS001980
View
Dmax
-
=
84
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002212
PGDB_C031991
PGDB_AS001980
View
Dmax
-
=
83
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002900
PGDB_C031975
PGDB_AS001980
View
Dmax
-
=
89
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003164
PGDB_C031992
PGDB_AS001980
View
Dmax
-
=
82
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003173
PGDB_C031962
PGDB_AS001980
View
Dmax
-
=
83
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003191
PGDB_C031953
PGDB_AS001980
View
Dmax
-
=
79
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003578
PGDB_C031982
PGDB_AS001980
View
Dmax
-
=
64
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003886
PGDB_C031987
PGDB_AS001980
View
Dmax
-
=
79
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003951
PGDB_C031973
PGDB_AS001980
View
Dmax
-
=
76
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A004111
PGDB_C031947
PGDB_AS001980
View
Dmax
-
=
69
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A004220
PGDB_C031978
PGDB_AS001980
View