Assay

PGDB_AS001984

System: cell_basedTarget: VAV1
Assay context summary

Assay context

77 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetVAV1
E3Not specified
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C032005
DC50-=2nM-—VAV1--WO2026119120A1PGDB_A000026PGDB_C032005PGDB_AS001984View
2D structure for PGDB_C032057
DC50-=4.2nM-—VAV1--WO2026119120A1PGDB_A000043PGDB_C032057PGDB_AS001984View
2D structure for PGDB_C024751
DC50-=4.7nM-—VAV1--WO2026119120A1PGDB_A000338PGDB_C024751PGDB_AS001984View
2D structure for PGDB_C032042
DC50-=3nM-—VAV1--WO2026119120A1PGDB_A000372PGDB_C032042PGDB_AS001984View
2D structure for PGDB_C009245
DC50-=5.9nM-—VAV1--WO2026119120A1PGDB_A000433PGDB_C009245PGDB_AS001984View
2D structure for PGDB_C032053
DC50-=1.1nM-—VAV1--WO2026119120A1PGDB_A000463PGDB_C032053PGDB_AS001984View
2D structure for PGDB_C032012
DC50-=42nM-—VAV1--WO2026119120A1PGDB_A000631PGDB_C032012PGDB_AS001984View
2D structure for PGDB_C032063
DC50-=11.1nM-—VAV1--WO2026119120A1PGDB_A000726PGDB_C032063PGDB_AS001984View
2D structure for PGDB_C032041
DC50-=2.3nM-—VAV1--WO2026119120A1PGDB_A000836PGDB_C032041PGDB_AS001984View
2D structure for PGDB_C024792
DC50-=4.8nM-—VAV1--WO2026119120A1PGDB_A001005PGDB_C024792PGDB_AS001984View
2D structure for PGDB_C032040
DC50-=5.8nM-—VAV1--WO2026119120A1PGDB_A001011PGDB_C032040PGDB_AS001984View
2D structure for PGDB_C032067
DC50-=2.7nM-—VAV1--WO2026119120A1PGDB_A001117PGDB_C032067PGDB_AS001984View
2D structure for PGDB_C032055
DC50-=1.9nM-—VAV1--WO2026119120A1PGDB_A001351PGDB_C032055PGDB_AS001984View
2D structure for PGDB_C032062
DC50-=5.6nM-—VAV1--WO2026119120A1PGDB_A001424PGDB_C032062PGDB_AS001984View
2D structure for PGDB_C032064
DC50-=13.9nM-—VAV1--WO2026119120A1PGDB_A001467PGDB_C032064PGDB_AS001984View
2D structure for PGDB_C032061
DC50-=7.3nM-—VAV1--WO2026119120A1PGDB_A001472PGDB_C032061PGDB_AS001984View
2D structure for PGDB_C032050
DC50-=10.2nM-—VAV1--WO2026119120A1PGDB_A001773PGDB_C032050PGDB_AS001984View
2D structure for PGDB_C032047
DC50-=4.4nM-—VAV1--WO2026119120A1PGDB_A001811PGDB_C032047PGDB_AS001984View
2D structure for PGDB_C032009
DC50-=13.8nM-—VAV1--WO2026119120A1PGDB_A001947PGDB_C032009PGDB_AS001984View
2D structure for PGDB_C032024
DC50-=1.8nM-—VAV1--WO2026119120A1PGDB_A002074PGDB_C032024PGDB_AS001984View
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