Assay context summary

Assay context

37 activity records
Activity compounds and values

Activity records

37 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031967
IC50-=3.8nM--CRBNGP5dWO2026114958A1PGDB_A000003PGDB_C031967PGDB_AS002003View
2D structure for PGDB_C031991
IC50-=2nM--CRBNGP5dWO2026114958A1PGDB_A000059PGDB_C031991PGDB_AS002003View
2D structure for PGDB_C031997
IC50-=6nM--CRBNGP5dWO2026114958A1PGDB_A000695PGDB_C031997PGDB_AS002003View
2D structure for PGDB_C031943
IC50-=1.5nM--CRBNGP5dWO2026114958A1PGDB_A001276PGDB_C031943PGDB_AS002003View
2D structure for PGDB_C031976
IC50-=5.4nM--CRBNGP5dWO2026114958A1PGDB_A001735PGDB_C031976PGDB_AS002003View
2D structure for PGDB_C031947
IC50-=5.2nM--CRBNGP5dWO2026114958A1PGDB_A002166PGDB_C031947PGDB_AS002003View
2D structure for PGDB_C031995
IC50-=2.5nM--CRBNGP5dWO2026114958A1PGDB_A002176PGDB_C031995PGDB_AS002003View
2D structure for PGDB_C031952
IC50-=3.9nM--CRBNGP5dWO2026114958A1PGDB_A002337PGDB_C031952PGDB_AS002003View
2D structure for PGDB_C031960
IC50-=1.8nM--CRBNGP5dWO2026114958A1PGDB_A002372PGDB_C031960PGDB_AS002003View
2D structure for PGDB_C031973
IC50-=1000nM--CRBNGP5dWO2026114958A1PGDB_A002648PGDB_C031973PGDB_AS002003View
2D structure for PGDB_C031989
IC50-=25.6nM--CRBNGP5dWO2026114958A1PGDB_A002898PGDB_C031989PGDB_AS002003View
2D structure for PGDB_C031988
IC50-=5.2nM--CRBNGP5dWO2026114958A1PGDB_A003088PGDB_C031988PGDB_AS002003View
2D structure for PGDB_C031970
IC50-=7.4nM--CRBNGP5dWO2026114958A1PGDB_A003674PGDB_C031970PGDB_AS002003View
2D structure for PGDB_C031942
IC50-=23.4nM--CRBNGP5dWO2026114958A1PGDB_A004402PGDB_C031942PGDB_AS002003View
2D structure for PGDB_C031949
IC50-=1.8nM--CRBNGP5dWO2026114958A1PGDB_A004723PGDB_C031949PGDB_AS002003View
2D structure for PGDB_C031941
IC50-=0.2nM--CRBNGP5dWO2026114958A1PGDB_A004942PGDB_C031941PGDB_AS002003View
2D structure for PGDB_C031993
IC50-=2.5nM--CRBNGP5dWO2026114958A1PGDB_A005006PGDB_C031993PGDB_AS002003View
2D structure for PGDB_C031985
IC50-=2.6nM--CRBNGP5dWO2026114958A1PGDB_A005133PGDB_C031985PGDB_AS002003View
2D structure for PGDB_C031990
IC50-=6.6nM--CRBNGP5dWO2026114958A1PGDB_A005139PGDB_C031990PGDB_AS002003View
2D structure for PGDB_C031976
IC50-=4.4nM--CRBNGP5dWO2026114958A1PGDB_A005412PGDB_C031976PGDB_AS002003View