Assay context summary

Assay context

35 activity records
Activity compounds and values

Activity records

35 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C003368
IC50-=8nM---MDA-MB-453WO2026007898A1PGDB_A009179PGDB_C003368PGDB_AS002028View
2D structure for PGDB_C003376
IC50-=1.2nM---MDA-MB-453WO2026007898A1PGDB_A009278PGDB_C003376PGDB_AS002028View
2D structure for PGDB_C003375
IC50-=1834nM---MDA-MB-453WO2026007898A1PGDB_A010585PGDB_C003375PGDB_AS002028View
2D structure for PGDB_C003385
IC50-=2nM---MDA-MB-453WO2026007898A1PGDB_A011614PGDB_C003385PGDB_AS002028View
2D structure for PGDB_C003388
IC50-=267nM---MDA-MB-453WO2026007898A1PGDB_A013277PGDB_C003388PGDB_AS002028View
2D structure for PGDB_C003372
IC50-=51nM---MDA-MB-453WO2026007898A1PGDB_A014408PGDB_C003372PGDB_AS002028View
2D structure for PGDB_C003367
IC50-=2nM---MDA-MB-453WO2026007898A1PGDB_A014982PGDB_C003367PGDB_AS002028View
2D structure for PGDB_C003391
IC50-=39nM---MDA-MB-453WO2026007898A1PGDB_A018125PGDB_C003391PGDB_AS002028View
2D structure for PGDB_C003380
IC50-=151nM---MDA-MB-453WO2026007898A1PGDB_A021331PGDB_C003380PGDB_AS002028View
2D structure for PGDB_C003390
IC50-=109nM---MDA-MB-453WO2026007898A1PGDB_A023331PGDB_C003390PGDB_AS002028View
2D structure for PGDB_C003374
IC50-=45nM---MDA-MB-453WO2026007898A1PGDB_A023492PGDB_C003374PGDB_AS002028View
2D structure for PGDB_C003383
IC50-=3nM---MDA-MB-453WO2026007898A1PGDB_A023742PGDB_C003383PGDB_AS002028View
2D structure for PGDB_C003393
IC50->10000nM---MDA-MB-453WO2026007898A1PGDB_A024614PGDB_C003393PGDB_AS002028View
2D structure for PGDB_C003370
IC50-=5nM---MDA-MB-453WO2026007898A1PGDB_A025695PGDB_C003370PGDB_AS002028View
2D structure for PGDB_C003396
IC50-=206nM---MDA-MB-453WO2026007898A1PGDB_A026564PGDB_C003396PGDB_AS002028View
2D structure for PGDB_C003371
IC50-=101nM---MDA-MB-453WO2026007898A1PGDB_A029085PGDB_C003371PGDB_AS002028View
2D structure for PGDB_C003369
IC50-=119nM---MDA-MB-453WO2026007898A1PGDB_A029944PGDB_C003369PGDB_AS002028View
2D structure for PGDB_C003389
IC50-=252nM---MDA-MB-453WO2026007898A1PGDB_A030404PGDB_C003389PGDB_AS002028View
2D structure for PGDB_C003379
IC50-=89nM---MDA-MB-453WO2026007898A1PGDB_A032449PGDB_C003379PGDB_AS002028View
2D structure for PGDB_C003381
IC50-=60nM---MDA-MB-453WO2026007898A1PGDB_A032734PGDB_C003381PGDB_AS002028View