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Compound
PGDB_C003380
6 activity records1 related patents
2D structure
CC(C)NCCOCCc1ccc(NC(=O)N[C@@H](C)c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 151 | nM | - | — | - | - | MDA-MB-453 | WO2026007898A1 | PGDB_A021331 | PGDB_C003380 | PGDB_AS002028 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF1 | - | - | WO2026007898A1 | PGDB_A035846 | PGDB_C003380 | PGDB_AS002166 | View |
| DC50 | - | = | 14.2 | nM | - | — | GSPT1 | - | - | WO2026007898A1 | PGDB_A039796 | PGDB_C003380 | PGDB_AS002374 | View |
| Selectivity index | IKZF3 | > | 704 | fold | - | — | - | - | - | WO2026007898A1 | PGDB_A040191 | PGDB_C003380 | PGDB_AS000375 | View |
| Selectivity index | IKZF1 | > | 704 | fold | - | — | - | - | - | WO2026007898A1 | PGDB_A048170 | PGDB_C003380 | PGDB_AS001314 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | - | WO2026007898A1 | PGDB_A064310 | PGDB_C003380 | PGDB_AS002393 | View |