Assay
PGDB_AS002039
System: biochemicalTarget: CRBN | DDB1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.08703 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A026330 | PGDB_C007378 | PGDB_AS002039 | View | |
| IC50 | - | = | 0.24971 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A031740 | PGDB_C007374 | PGDB_AS002039 | View | |
| IC50 | - | = | 0.2906 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A044273 | PGDB_C007377 | PGDB_AS002039 | View | |
| IC50 | - | = | 0.30892 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A048467 | PGDB_C007379 | PGDB_AS002039 | View | |
| IC50 | - | = | 0.1291 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A064569 | PGDB_C007376 | PGDB_AS002039 | View | |
| IC50 | - | = | 0.08729 | uM | - | — | CRBN | CRBN | - | CN121378270A | PGDB_A073274 | PGDB_C007375 | PGDB_AS002039 | View |