Assay
PGDB_AS002069
System: cell_basedCell line: NCI-H1299
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.12 | nM | - | — | GSPT1 | - | NCI-H1299 | CN120365257A | PGDB_A045429 | PGDB_C000737 | PGDB_AS002069 | View | |
| IC50 | - | = | 24.34 | nM | - | — | GSPT1 | - | NCI-H1299 | CN120365257A | PGDB_A045888 | PGDB_C000739 | PGDB_AS002069 | View | |
| IC50 | - | = | 7.37 | nM | - | — | GSPT1 | - | NCI-H1299 | CN120365257A | PGDB_A061391 | PGDB_C000735 | PGDB_AS002069 | View | |
| IC50 | - | = | 9.41 | nM | - | — | GSPT1 | - | NCI-H1299 | CN120365257A | PGDB_A065620 | PGDB_C000736 | PGDB_AS002069 | View | |
| IC50 | - | = | 0.47 | nM | - | — | GSPT1 | - | NCI-H1299 | CN120365257A | PGDB_A067133 | PGDB_C000738 | PGDB_AS002069 | View |