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SIMM · NJU
Assay
PGDB_AS002112
System: cell_based
Target: IKZF2
Cell line: 293GT
Assay context summary
Assay context
150 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
Target
IKZF2
E3
Not specified
Cell line
293GT
Organism
Homo sapiens
Detection target
protein_degradation
Activity compounds and values
Activity records
150 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
55.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007048
PGDB_C022664
PGDB_AS002112
View
% Degradation
-
=
60.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007230
PGDB_C022669
PGDB_AS002112
View
% Degradation
-
=
60.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007471
PGDB_C022735
PGDB_AS002112
View
% Degradation
-
=
50.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007536
PGDB_C022645
PGDB_AS002112
View
% Degradation
-
=
70.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007588
PGDB_C022694
PGDB_AS002112
View
% Degradation
-
=
50.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A007938
PGDB_C022742
PGDB_AS002112
View
% Degradation
-
=
80.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A008190
PGDB_C022746
PGDB_AS002112
View
% Degradation
-
=
5.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A008579
PGDB_C022702
PGDB_AS002112
View
% Degradation
-
=
50.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A008617
PGDB_C022649
PGDB_AS002112
View
% Degradation
-
=
70.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A008804
PGDB_C022732
PGDB_AS002112
View
% Degradation
-
=
50.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A008875
PGDB_C022681
PGDB_AS002112
View
% Degradation
-
=
80.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A009010
PGDB_C022704
PGDB_AS002112
View
% Degradation
-
=
75.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A009106
PGDB_C022695
PGDB_AS002112
View
% Degradation
-
=
80.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A009228
PGDB_C022680
PGDB_AS002112
View
% Degradation
-
=
75.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A011165
PGDB_C022654
PGDB_AS002112
View
% Degradation
-
=
45.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A011865
PGDB_C022640
PGDB_AS002112
View
% Degradation
-
=
40.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A012200
PGDB_C022769
PGDB_AS002112
View
% Degradation
-
=
60.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A012990
PGDB_C022763
PGDB_AS002112
View
% Degradation
-
=
50.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A013443
PGDB_C022698
PGDB_AS002112
View
% Degradation
-
=
40.0
%
10 uM
24 h
-
-
293GT
CN111051298A
PGDB_A013808
PGDB_C022677
PGDB_AS002112
View