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N#CCc1ccc(CN2CCC(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 80.0 | % | 10 uM | 24 h | - | - | 293GT | CN111051298A | PGDB_A009228 | PGDB_C022680 | PGDB_AS002112 | View | |
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A013005 | PGDB_C022680 | PGDB_AS002316 | View | |
| EC50 | - | > | 30.0 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A045557 | PGDB_C022680 | PGDB_AS000334 | View | |
| EC50 | - | = | 0.009 | uM | - | — | - | - | 293GT | CN111051298A | PGDB_A051621 | PGDB_C022680 | PGDB_AS001169 | View |