Assay context summary

Assay context

50 activity records
Activity compounds and values

Activity records

50 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C003233
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A007277PGDB_C003233PGDB_AS002114View
2D structure for PGDB_C003222
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A011435PGDB_C003222PGDB_AS002114View
2D structure for PGDB_C003237
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A012263PGDB_C003237PGDB_AS002114View
2D structure for PGDB_C003249
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A013037PGDB_C003249PGDB_AS002114View
2D structure for PGDB_C003236
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A015572PGDB_C003236PGDB_AS002114View
2D structure for PGDB_C003238
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A019084PGDB_C003238PGDB_AS002114View
2D structure for PGDB_C003223
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A019248PGDB_C003223PGDB_AS002114View
2D structure for PGDB_C003229
IC50-=100-1000nM-GSPT1-KG-1WO2024222918A1PGDB_A023217PGDB_C003229PGDB_AS002114View
2D structure for PGDB_C003256
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A024016PGDB_C003256PGDB_AS002114View
2D structure for PGDB_C003224
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A024264PGDB_C003224PGDB_AS002114View
2D structure for PGDB_C003246
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A024584PGDB_C003246PGDB_AS002114View
2D structure for PGDB_C003265
IC50-<1nM-GSPT1-KG-1WO2024222918A1PGDB_A024929PGDB_C003265PGDB_AS002114View
2D structure for PGDB_C003251
IC50->=1000nM-GSPT1-KG-1WO2024222918A1PGDB_A027040PGDB_C003251PGDB_AS002114View
2D structure for PGDB_C003250
IC50->=1000nM-GSPT1-KG-1WO2024222918A1PGDB_A027709PGDB_C003250PGDB_AS002114View
2D structure for PGDB_C003247
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A027769PGDB_C003247PGDB_AS002114View
2D structure for PGDB_C003225
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A028450PGDB_C003225PGDB_AS002114View
2D structure for PGDB_C003226
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A028728PGDB_C003226PGDB_AS002114View
2D structure for PGDB_C003266
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A030665PGDB_C003266PGDB_AS002114View
2D structure for PGDB_C003239
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A032597PGDB_C003239PGDB_AS002114View
2D structure for PGDB_C003259
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A033456PGDB_C003259PGDB_AS002114View