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SIMM · NJU
Assay
PGDB_AS002165
System: cell_based
Target: NEK7
Assay context summary
Assay context
212 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
NEK7
E3
CRBN
Activity compounds and values
Activity records
212 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A007062
PGDB_C020324
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A007786
PGDB_C020440
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A007964
PGDB_C020405
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008148
PGDB_C020338
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008217
PGDB_C020293
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008304
PGDB_C020422
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008325
PGDB_C020414
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008361
PGDB_C016360
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008870
PGDB_C020435
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A009188
PGDB_C020296
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A009845
PGDB_C020451
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A009978
PGDB_C020339
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A010391
PGDB_C020333
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A010656
PGDB_C026263
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A010845
PGDB_C020424
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A012421
PGDB_C020364
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A012650
PGDB_C026288
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A012709
PGDB_C020176
PGDB_AS002165
View
Dmax
-
>
75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A013310
PGDB_C026233
PGDB_AS002165
View
Dmax
-
=
50-75
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A013445
PGDB_C020450
PGDB_AS002165
View