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SIMM · NJU
Assay
PGDB_AS002224
System: cell_based
Assay context summary
Assay context
19 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
CRBN
Activity compounds and values
Activity records
19 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
95
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A014512
PGDB_C020442
PGDB_AS002224
View
Dmax
-
=
68
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A022511
PGDB_C020444
PGDB_AS002224
View
Dmax
-
=
70
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A029232
PGDB_C020446
PGDB_AS002224
View
Dmax
-
=
79
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A030133
PGDB_C020449
PGDB_AS002224
View
Dmax
-
=
90
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A030964
PGDB_C020436
PGDB_AS002224
View
Dmax
-
=
61
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A033987
PGDB_C020448
PGDB_AS002224
View
Dmax
-
=
57
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A035146
PGDB_C020445
PGDB_AS002224
View
Dmax
-
=
60
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A039277
PGDB_C020453
PGDB_AS002224
View
Dmax
-
=
61
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A044886
PGDB_C020450
PGDB_AS002224
View
Dmax
-
=
82
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A049471
PGDB_C020439
PGDB_AS002224
View
Dmax
-
=
71
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A052492
PGDB_C020451
PGDB_AS002224
View
Dmax
-
=
54
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A053658
PGDB_C020452
PGDB_AS002224
View
Dmax
-
=
88
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A054399
PGDB_C020435
PGDB_AS002224
View
Dmax
-
=
3
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057782
PGDB_C020447
PGDB_AS002224
View
Dmax
-
=
78
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057828
PGDB_C020455
PGDB_AS002224
View
Dmax
-
=
94
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057954
PGDB_C020440
PGDB_AS002224
View
Dmax
-
=
88
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A059033
PGDB_C020438
PGDB_AS002224
View
Dmax
-
=
68
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A063518
PGDB_C020437
PGDB_AS002224
View
Dmax
-
=
67
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A073006
PGDB_C020454
PGDB_AS002224
View