Assay
PGDB_AS002362
System: cell_basedCell line: U937
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A014025 | PGDB_C003221 | PGDB_AS002362 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A016725 | PGDB_C000059 | PGDB_AS002362 | View | |
| IC50 | - | = | 1-10 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A036335 | PGDB_C003219 | PGDB_AS002362 | View | |
| IC50 | - | = | 1-10 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A064163 | PGDB_C003262 | PGDB_AS002362 | View | |
| IC50 | - | = | 1-10 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A066008 | PGDB_C003237 | PGDB_AS002362 | View | |
| IC50 | - | >= | 1000 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A070111 | PGDB_C003267 | PGDB_AS002362 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A074663 | PGDB_C003266 | PGDB_AS002362 | View | |
| IC50 | - | = | 1-10 | nM | - | — | GSPT1 | - | U937 | WO2024222918A1 | PGDB_A076929 | PGDB_C003265 | PGDB_AS002362 | View |