Assay

PGDB_AS002373

System: cell_basedCell line: THP-1
Assay context summary

Assay context

65 activity records
Assay familyviability
Systemcell_based
ReadoutGI50
E3Not specified
Cell lineTHP-1
OrganismHomo sapiens
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

65 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C012006
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A010301PGDB_C012006PGDB_AS002373View
2D structure for PGDB_C012014
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A010539PGDB_C012014PGDB_AS002373View
2D structure for PGDB_C011998
GI50-<1000nM-—CCNK-THP-1WO2025245472A1PGDB_A010681PGDB_C011998PGDB_AS002373View
2D structure for PGDB_C012028
GI50-<1000nM-—CCNK-THP-1WO2025245472A1PGDB_A011656PGDB_C012028PGDB_AS002373View
2D structure for PGDB_C012038
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A014609PGDB_C012038PGDB_AS002373View
2D structure for PGDB_C012040
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A016359PGDB_C012040PGDB_AS002373View
2D structure for PGDB_C012005
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A018300PGDB_C012005PGDB_AS002373View
2D structure for PGDB_C012010
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A019614PGDB_C012010PGDB_AS002373View
2D structure for PGDB_C012016
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A020785PGDB_C012016PGDB_AS002373View
2D structure for PGDB_C012013
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A020877PGDB_C012013PGDB_AS002373View
2D structure for PGDB_C012030
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A022023PGDB_C012030PGDB_AS002373View
2D structure for PGDB_C012012
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A022082PGDB_C012012PGDB_AS002373View
2D structure for PGDB_C011999
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A022722PGDB_C011999PGDB_AS002373View
2D structure for PGDB_C011995
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A023956PGDB_C011995PGDB_AS002373View
2D structure for PGDB_C012018
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A024718PGDB_C012018PGDB_AS002373View
2D structure for PGDB_C012001
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A024958PGDB_C012001PGDB_AS002373View
2D structure for PGDB_C012037
GI50-<1000nM-—CCNK-THP-1WO2025245472A1PGDB_A024994PGDB_C012037PGDB_AS002373View
2D structure for PGDB_C011975
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A026697PGDB_C011975PGDB_AS002373View
2D structure for PGDB_C012020
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A027580PGDB_C012020PGDB_AS002373View
2D structure for PGDB_C012003
GI50->3000nM-—CCNK-THP-1WO2025245472A1PGDB_A028399PGDB_C012003PGDB_AS002373View
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