Assay
PGDB_AS002469
System: cell_basedCell line: HEK293T
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.024 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A007882 | PGDB_C000380 | PGDB_AS002469 | View | |
| DC50 | - | > | 30 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A008252 | PGDB_C000383 | PGDB_AS002469 | View | |
| DC50 | - | > | 30 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A011098 | PGDB_C000382 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A031102 | PGDB_C000385 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.0005 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A031427 | PGDB_C000389 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.292 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A044816 | PGDB_C000384 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.006 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A047204 | PGDB_C000381 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.005 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A059796 | PGDB_C000387 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A063787 | PGDB_C000386 | PGDB_AS002469 | View | |
| DC50 | - | = | 0.005 | uM | - | — | IKZF2 | - | HEK293T | US20230265071A1 | PGDB_A070519 | PGDB_C000388 | PGDB_AS002469 | View |